A High-Throughput Dose-Response Cellular Thermal Shift Assay for Rapid Screening of Drug Target Engagement in Living Cells, Exemplified Using SMYD3 and IDO1

Autor: McNulty, Dean E. **, Bonnette, William G., Qi, Hongwei, Wang, Liping, Ho, Thau F., Waszkiewicz, Anna, Kallal, Lorena A., Nagarajan, Raman P., Stern, Melissa, Quinn, Amy M., Creasy, Caretha L., Su, Dai-Shi, Graves, Alan P., Annan, Roland S., Sweitzer, Sharon M., Holbert, Marc A. *
Zdroj: In SLAS Discovery January 2018 23(1):34-46
Databáze: ScienceDirect