BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability

Autor:	Jennings, Laura E., Schiedel, Matthias, Hewings, David S., Picaud, Sarah, Laurin, Corentine M.C., Bruno, Paul A., Bluck, Joseph P., Scorah, Amy R., See, Larissa, Reynolds, Jessica K., Moroglu, Mustafa, Mistry, Ishna N., Hicks, Amy, Guzanov, Pavel, Clayton, James, Evans, Charles N.G., Stazi, Giulia, Biggin, Philip C., Mapp, Anna K., Hammond, Ester M., Humphreys, Philip G., Filippakopoulos, Panagis, Conway, Stuart J.
Zdroj:	In Bioorganic & Medicinal Chemistry 15 July 2018 26(11):2937-2957
Databáze:	ScienceDirect
Externí odkaz:	Zobrazit plný text záznamu Full Text from ScienceDirect