Identification of 4-benzylamino-2-[(4-morpholin-4-ylphenyl)amino]pyrimidine-5-carboxamide derivatives as potent and orally bioavailable STAT6 inhibitors

Autor: Nagashima, Shinya, Nagata, Hiroshi, Iwata, Masahiro, Yokota, Masaki, Moritomo, Hiroyuki, Orita, Masaya, Kuromitsu, Sadao, Koakutsu, Akiko, Ohga, Keiko, Takeuchi, Makoto, Ohta, Mitsuaki, Tsukamoto, Shin-ichi
Zdroj: In Bioorganic & Medicinal Chemistry 2008 16(13):6509-6521
Databáze: ScienceDirect