Discovery of 1-[2-(1-methyl-1H-pyrazol-5-yl)-[1,2,4]triazolo[1,5-a]pyridin-6-yl]-3-(pyridin-4-ylmethyl)urea as a potent NAMPT (nicotinamide phosphoribosyltransferase) activator with attenuated CYP inhibition

Autor: Akiu, Mayuko, Tsuji, Takashi, Sogawa, Yoshitaka, Terayama, Koji, Yokoyama, Mika, Tanaka, Jun, Asano, Daigo, Sakurai, Ken, Sergienko, Eduard, Sessions, E. Hampton, Gardell, Stephen J., Pinkerton, Anthony B., Nakamura, Tsuyoshi
Zdroj: In Bioorganic & Medicinal Chemistry Letters 1 July 2021 43
Databáze: ScienceDirect