Discovery of novel histone lysine methyltransferase G9a/GLP (EHMT2/1) inhibitors: Design, synthesis, and structure-activity relationships of 2,4-diamino-6-methylpyrimidines

Autor: Katayama, Katsushi, Ishii, Ken, Tsuda, Eisuke, Yotsumoto, Keiichi, Hiramoto, Kumiko, Suzuki, Makoto, Yasumatsu, Isao, Igarashi, Wataru, Torihata, Munefumi, Ishiyama, Takashi, Katagiri, Takahiro
Zdroj: In Bioorganic & Medicinal Chemistry Letters 15 October 2020 30(20)
Databáze: ScienceDirect