Discovery of novel quinoline sulphonamide derivatives as potent, selective and orally active RORγ inverse agonists

Autor: Amaudrut, Jérôme, Argiriadi, Maria A., Barth, Martine, Breinlinger, Eric C., Bressac, Didier, Broqua, Pierre, Calderwood, David J., Chatar, Mohamed, Cusack, Kevin P., Gauld, Stephen B., Jacquet, Sébastien, Kamath, Rajesh V., Kort, Michael E., Lepais, Valérie, Luccarini, Jean-Michel, Masson, Philippe, Montalbetti, Christian, Mounier, Laurent, Potin, Dominique, Poupardin, Olivia, Rouaud, Sylvie, Spitzer, Luc, Wallace, Craig D.
Zdroj: In Bioorganic & Medicinal Chemistry Letters 15 July 2019 29(14):1799-1806
Databáze: ScienceDirect
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