Discovery of a novel 2,4-dimethylquinoline-6-carboxamide M4 positive allosteric modulator (PAM) chemotype via scaffold hopping

Autor: Long, Madeline F., Engers, Julie L., Chang, Sichen, Zhan, Xiaoyan, Weiner, Rebecca L., Luscombe, Vincent B., Rodriguez, Alice L., Cho, Hyekyung P., Niswender, Colleen M., Bridges, Thomas M., Conn, P. Jeffrey, Engers, Darren W., Lindsley, Craig W.
Zdroj: In Bioorganic & Medicinal Chemistry Letters 15 November 2017 27(22):4999-5001
Databáze: ScienceDirect