Discovery of a novel 2,4-dimethylquinoline-6-carboxamide M4 positive allosteric modulator (PAM) chemotype via scaffold hopping
Autor: | Long, Madeline F., Engers, Julie L., Chang, Sichen, Zhan, Xiaoyan, Weiner, Rebecca L., Luscombe, Vincent B., Rodriguez, Alice L., Cho, Hyekyung P., Niswender, Colleen M., Bridges, Thomas M., Conn, P. Jeffrey, Engers, Darren W., Lindsley, Craig W. |
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Zdroj: | In Bioorganic & Medicinal Chemistry Letters 15 November 2017 27(22):4999-5001 |
Databáze: | ScienceDirect |
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