Discovery of a biarylamide series of potent, state-dependent NaV1.7 inhibitors

Autor: Schenkel, Laurie B., DiMauro, Erin F., Nguyen, Hanh N., Chakka, Nagasree, Du, Bingfan, Foti, Robert S., Guzman-Perez, Angel, Jarosh, Michael, La, Daniel S., Ligutti, Joseph, Milgram, Benjamin C., Moyer, Bryan D., Peterson, Emily A., Roberts, John, Yu, Violeta L., Weiss, Matthew M.
Zdroj: In Bioorganic & Medicinal Chemistry Letters 15 August 2017 27(16):3817-3824
Databáze: ScienceDirect