Discovery of oxa-sultams as RORc inverse agonists showing reduced lipophilicity, improved selectivity and favorable ADME properties
| Autor: | René, Olivier, Fauber, Benjamin P., Barnard, Adrian, Chapman, Kerry, Deng, Yuzhong, Eidenschenk, Céline, Everett, Christine, Gobbi, Alberto, Johnson, Adam R., La, Hank, Norman, Maxine, Salmon, Gary, Summerhill, Susan, Wong, Harvey |
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| Zdroj: | In Bioorganic & Medicinal Chemistry Letters 15 September 2016 26(18):4455-4461 |
| Databáze: | ScienceDirect |
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