Design of selective PI3Kα inhibitors starting from a promiscuous pan kinase scaffold

Autor: Barlaam, Bernard, Cosulich, Sabina, Fitzek, Martina, Green, Stephen, Harris, Craig S., Hudson, Kevin, Lambert-van der Brempt, Christine, Ouvry, Gilles, Page, Ken, Ruston, Linette, Ward, Lara, Delouvrié, Bénédicte
Zdroj: In Bioorganic & Medicinal Chemistry Letters 1 July 2015 25(13):2679-2685
Databáze: ScienceDirect