Discovery of 9-(1-anilinoethyl)-2-morpholino-4-oxo-pyrido[1,2-a]pyrimidine-7-carboxamides as PI3Kβ/δ inhibitors for the treatment of PTEN-deficient tumours

Autor: Barlaam, Bernard, Cosulich, Sabina, Degorce, Sébastien, Fitzek, Martina, Giordanetto, Fabrizio, Green, Stephen, Inghardt, Tord, Hennequin, Laurent, Hancox, Urs, Lambert-van der Brempt, Christine, Morgentin, Rémy, Pass, Sarah, Plé, Patrick, Saleh, Twana, Ward, Lara
Zdroj: In Bioorganic & Medicinal Chemistry Letters 15 August 2014 24(16):3928-3935
Databáze: ScienceDirect