Discovery of triazolopyrimidine-based PDE8B inhibitors: Exceptionally ligand-efficient and lipophilic ligand-efficient compounds for the treatment of diabetes
Autor: | DeNinno, Michael P., Wright, Stephen W., Etienne, John B., Olson, Thanh V., Rocke, Benjamin N., Corbett, Jeffrey W., Kung, Daniel W., DiRico, Kenneth J., Andrews, Kim M., Millham, Michele L., Parker, Janice C., Esler, William, van Volkenburg, Maria, Boyer, David D., Houseknecht, Karen L., Doran, Shawn D. |
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Zdroj: | In Bioorganic & Medicinal Chemistry Letters 1 September 2012 22(17):5721-5726 |
Databáze: | ScienceDirect |
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