Structure-based library design and the discovery of a potent and selective mast cell β-tryptase inhibitor as an oral therapeutic agent

Autor: Liang, Guyan, Aldous, Suzanne, Merriman, Gregory, Levell, Julian, Pribish, James, Cairns, Jennifer, Chen, Xin, Maignan, Sebastien, Mathieu, Magali, Tsay, Joseph, Sides, Keith, Rebello, Sam, Whitely, Brian, Morize, Isabelle, Pauls, Henry W.
Zdroj: In Bioorganic & Medicinal Chemistry Letters 15 January 2012 22(2):1049-1054
Databáze: ScienceDirect