Discovery of pyrrolo[2,1- f][1,2,4]triazine C6-ketones as potent, orally active p38α MAP kinase inhibitors
Autor: | Dyckman, Alaric J., Li, Tianle, Pitt, Sidney, Zhang, Rosemary, Shen, Ding Ren, McIntyre, Kim W., Gillooly, Kathleen M., Shuster, David J., Doweyko, Arthur M., Sack, John S., Kish, Kevin, Kiefer, Susan E., Newitt, John A., Zhang, Hongjian, Marathe, Punit H., McKinnon, Murray, Barrish, Joel C., Dodd, John H., Schieven, Gary L., Leftheris, Katerina |
---|---|
Zdroj: | In Bioorganic & Medicinal Chemistry Letters 2011 21(15):4633-4637 |
Databáze: | ScienceDirect |
Externí odkaz: |