Design of novel and potent cPLA 2α inhibitors containing an α-methyl-2-ketothiazole as a metabolically stable serine trap

Autor: Mete, Antonio, Andrews, Glen, Bernstein, Mike, Connolly, Stephen, Hartopp, Paul, Jackson, Clive G., Lewis, Richard, Martin, Iain, Murray, David, Riley, Rob, Robinson, David H., Smith, Gill M., Wells, Edward, Withnall, W. John
Zdroj: In Bioorganic & Medicinal Chemistry Letters 2011 21(10):3128-3133
Databáze: ScienceDirect