Hit-to-lead optimization of a series of carboxamides of ethyl 2-amino-4-phenylthiazole-5-carboxylates as novel adenosine A 2A receptor antagonists

Autor: Sams, Anette Graven, Mikkelsen, Gitte Kobberøe, Larsen, Mogens, Torup, Lars, Brennum, Lise Tøttrup, Schrøder, Tenna Juul, Bang-Andersen, Benny
Zdroj: In Bioorganic & Medicinal Chemistry Letters 2010 20(17):5241-5244
Databáze: ScienceDirect