Potent, selective, orally bioavailable inhibitors of tumor necrosis factor-α converting enzyme (TACE): Discovery of indole, benzofuran, imidazopyridine and pyrazolopyridine P1′ substituents

Autor: Lu, Zhonghui, Ott, Gregory R., Anand, Rajan, Liu, Rui-Qin, Covington, Maryanne B., Vaddi, Krishna, Qian, Mingxin, Newton, Robert C., Christ, David D., Trzaskos, James, Duan, James J.-W.
Zdroj: In Bioorganic & Medicinal Chemistry Letters 2008 18(6):1958-1962
Databáze: ScienceDirect