Discovery of 3-OH-3-methylpipecolic hydroxamates: Potent orally active inhibitors of aggrecanase and MMP-13

Autor: Noe, Mark C., Natarajan, Vijayalakshmi, Snow, Sheri L., Wolf-Gouveia, Lilli A., Mitchell, Peter G., Lopresti-Morrow, Lori, Reeves, Lisa M., Yocum, Sue A., Otterness, Ivan, Bliven, Marcia A., Carty, Thomas J., Barberia, John T., Sweeney, Francis J., Liras, Jennifer L., Vaughn, Marcie
Zdroj: In Bioorganic & Medicinal Chemistry Letters 2005 15(14):3385-3388
Databáze: ScienceDirect