Solubility-driven optimization of benzothiopyranone salts leading to a preclinical candidate with improved pharmacokinetic properties and activity against Mycobacterium tuberculosis

Autor: Li, Peng, Guo, Kaijing, Fu, Lei, Wang, Bin, Zhang, Baoxi, Gong, Ningbo, Lu, Yang, Ma, Chen, Huang, Haihong, Lu, Yu, Li, Gang
Zdroj: In European Journal of Medicinal Chemistry 15 January 2023 246
Databáze: ScienceDirect