Synthesis, bioconversion, pharmacokinetic and pharmacodynamic evaluation of N-isopropyl-oxy-carbonyloxymethyl prodrugs of CZh-226, a potent and selective PAK4 inhibitor
Autor: | Guo, Jing, Wang, Tingting, Wu, Tianxiao, Zhang, Kehan, Yin, Wenbo, Zhu, Mingyue, Pang, Yu, Hao, Chenzhou, He, Zhonggui, Cheng, Maosheng, Liu, Yang, Zheng, Jiang, Gu, Jingkai, Zhao, Dongmei |
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Zdroj: | In European Journal of Medicinal Chemistry 15 January 2020 186 |
Databáze: | ScienceDirect |
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