Discovery and optimization of 1-(1H-indol-1-yl)ethanone derivatives as CBP/EP300 bromodomain inhibitors for the treatment of castration-resistant prostate cancer
| Autor: | Xiang, Qiuping, Wang, Chao, Zhang, Yan, Xue, Xiaoqian, Song, Ming, Zhang, Cheng, Li, Chenchang, Wu, Chun, Li, Kuai, Hui, Xiaoyan, Zhou, Yulai, Smaill, Jeff B., Patterson, Adam V., Wu, Donghai, Ding, Ke, Xu, Yong |
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| Zdroj: | In European Journal of Medicinal Chemistry 10 March 2018 147:238-252 |
| Databáze: | ScienceDirect |
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