Structure-activity studies on N-Substituted tranylcypromine derivatives lead to selective inhibitors of lysine specific demethylase 1 (LSD1) and potent inducers of leukemic cell differentiation

Autor: Schulz-Fincke, Johannes, Hau, Mirjam, Barth, Jessica, Robaa, Dina, Willmann, Dominica, Kürner, Andreas, Haas, Julian, Greve, Gabriele, Haydn, Tinka, Fulda, Simone, Lübbert, Michael, Lüdeke, Steffen, Berg, Tobias, Sippl, Wolfgang, Schüle, Roland, Jung, Manfred
Zdroj: In European Journal of Medicinal Chemistry 20 January 2018 144:52-67
Databáze: ScienceDirect