Discovery, mechanism and metabolism studies of 2,3-difluorophenyl-linker-containing PARP1 inhibitors with enhanced in vivo efficacy for cancer therapy

Autor: Chen, Wenhua, Guo, Ne, Qi, Minghui, Dai, Haiying, Hong, Minghuang, Guan, Longfei, Huan, Xiajuan, Song, Shanshan, He, Jinxue, Wang, Yingqing, Xi, Yong, Yang, Xinying, Shen, Yanyan, Su, Yi, Sun, Yiming, Gao, Yinglei, Chen, Yi, Ding, Jian, Tang, Yun, Ren, Guobin, Miao, Zehong, Li, Jian
Zdroj: In European Journal of Medicinal Chemistry 29 September 2017 138:514-531
Databáze: ScienceDirect