Discovery of a series of dihydroquinoxalin-2(1H)-ones as selective BET inhibitors from a dual PLK1-BRD4 inhibitor

Autor: Hu, Jianping, Wang, Yingqing, Li, Yanlian, Xu, Lin, Cao, Danyan, Song, ShanShan, Damaneh, Mohammadali Soleimani, Wang, Xin, Meng, Tao, Chen, Yue-Lei, Shen, Jingkang, Miao, Zehong, Xiong, Bing
Zdroj: In European Journal of Medicinal Chemistry 8 September 2017 137:176-195
Databáze: ScienceDirect