X-ray crystallography study and optimization of novel benzothiophene analogs as potent selective estrogen receptor covalent antagonists (SERCAs) with improved potency and safety profiles

Autor: Bai, Chengfeng, Lv, Yang, Xiong, Shuangshuang, Wu, Shuangjie, Qi, Lin, Ren, Shengnan, Zhu, Meiqi, Dong, Haijuan, Shen, Hongtao, Li, Zhaoxing, Zhu, Yinxue, Ye, Hui, Hao, Haiping, Xiao, Yibei, Xiang, Hua, Luo, Guoshun
Zdroj: In Bioorganic Chemistry December 2023 141
Databáze: ScienceDirect