A Point Mutation That Confers Constitutive Activity to CXCR4 Reveals That T140 Is an Inverse Agonist and That AMD3100 and ALX40-4C Are Weak Partial Agonists

Autor: Zhang, Wen-bo ‡, §, ¶, Navenot, Jean-Marc ‡, §, ‖, Haribabu, Bodduluri , Tamamura, Hirokazu **, Hiramatu, Kenichi **, Omagari, Akane **, Pei, Gang , Manfredi, John P. §§, Fujii, Nobutaka **, Broach, James R. ¶¶, Peiper, Stephen C. ‡, 166, ‖
Zdroj: In Journal of Biological Chemistry 5 July 2002 277(27):24515-24521
Databáze: ScienceDirect