Mechanism for aromatase inactivation by a suicide substrate, androst-4-ene-3,6,17-trione: The 4β,5β-epoxy-19-oxo derivative as a reactive electrophile irreversibly binding to the active site

Autor: Numazawa, Mitsuteru, Mutsumi, Ayako, Tachibana, Mii
Zdroj: In Biochemical Pharmacology 1996 52(8):1253-1259
Databáze: ScienceDirect