Discovery and hit-to-lead evaluation of piperazine amides as selective, state-dependent Na

Autor:	Sparling, Brian A., Yi, S., Able, J., Bregman, H., DiMauro, Erin F., Foti, R. S., Gao, H., Guzman-Perez, A., Huang, H., Jarosh, M., Kornecook, T., Ligutti, J., Milgram, B. C., Moyer, B. D., Youngblood, B., Yu, V. L., Weiss, M. M.
Rok vydání:	2016
Předmět:	Chemistry
Zdroj:	MedChemComm. 8(4)
ISSN:	2040-2503
Popis:	Optimization of a screening hit led to the identification of NaV1.7 inhibitors with a desirable balance of properties.
Databáze:	OpenAIRE
Externí odkaz:	https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::f41ba3418e04c8c2792a5558d5f99e56 https://pubmed.ncbi.nlm.nih.gov/30108793 Zobrazit plný text záznamu