2,5-Diketopiperidine derivatives as non-peptide ligands for cholecystokinin receptors
Autor: | R G, González-Muñiz, M J, Domínguez, R, Herranz, M T, García-López, S J, Ballaz, A, Fortuño, J, Del Río |
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Rok vydání: | 1997 |
Předmět: | |
Zdroj: | Farmaco (Societa chimica italiana : 1989). 52(4) |
ISSN: | 0014-827X |
Popis: | Easily accessible 2,5-diketopiperidines have been used as templates for the construction of Trp-Phe and Trp-Asp-Phe-NH2 mimics. The cycle [L-Trp psi[COCH2]-L-Phe] analogue 1a has shown to possess significant and selective affinity for CCKA receptors. |
Databáze: | OpenAIRE |
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