Direct Arylation of Benzo[b]furan and Other Benzo-Fused Heterocycles

Autor:	Dao-Huy, Toan, Haider, Maximilian, Glatz, Fabian, Schnürch, Michael, Mihovilovic, Marko D
Jazyk:	angličtina
Rok vydání:	2014
Předmět:	Regioselectivity Synthetic methods Concerted metal deprotonation C–H activation Full Papers Arylation Fused-ring systems Palladium
Zdroj:	European Journal of Organic Chemistry
ISSN:	1099-0690 1434-193X
Popis:	The direct arylation of benzo[b]furan, benzo[b]thiophene, and indole has been studied by using aromatic bromides as the aryl source. The protocol employing common reagents and a Pd catalyst has led to the regioselective arylation of these heterocycles at the 2-position. A range of functional groups were tolerated, providing quick access to a variety of arylated benzo-fused heterocycles that would be accessible more elaborately using classical synthetic strategies. This is the first systematic study of the direct arylation of benzo[b]furan.
Databáze:	OpenAIRE
Externí odkaz:	https://explore.openaire.eu/search/publication?articleId=pmid________::7d4c95413c3759b0363e10b104c53a6a http://europepmc.org/articles/PMC4502765 Zobrazit plný text záznamu Plný text ve formátu PDF Plný text ve formátu HTML
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