The discovery of Arylex™ active and Rinskor™ active: Two novel auxin herbicides
| Autor: | Buysse Ann M, Thomas L. Siddall, Lowe Christian T, Brewster William, Lo William C, Terry William Balko, Roger E. Gast, Gregory T. Whiteker, Epp Jeffrey B, John F. Daeuble, Nicholas M. Irvine, Monte Weimer, Renard Antonio Green, John S. Richburg, Satchivi Norbert M, Webster Jeffery, James M. Renga, Carla N. Yerkes, James Melvin Ruiz, Anita Lenora Alexander, Kristy Bryan, Paul R. Schmitzer, Stephen Craig Fields |
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| Rok vydání: | 2015 |
| Předmět: |
0106 biological sciences
Mecoprop Clinical Biochemistry Pharmaceutical Science Picloram 01 natural sciences Biochemistry MCPA chemistry.chemical_compound Structure-Activity Relationship Drug Discovery Aminopyralid Quinclorac Molecular Biology Fluroxypyr Indoleacetic Acids Herbicides Organic Chemistry Oryza 04 agricultural and veterinary sciences Clopyralid chemistry Agronomy 040103 agronomy & agriculture 0401 agriculture forestry and fisheries Molecular Medicine Aminocyclopyrachlor Edible Grain 010606 plant biology & botany |
| Zdroj: | Bioorganicmedicinal chemistry. 24(3) |
| ISSN: | 1464-3391 |
| Popis: | Multiple classes of commercially important auxin herbicides have been discovered since the 1940s including the aryloxyacetates (2,4-D, MCPA, dichlorprop, mecoprop, triclopyr, and fluroxypyr), the benzoates (dicamba), the quinoline-2-carboxylates (quinclorac and quinmerac), the pyrimidine-4-carboxylates (aminocyclopyrachlor), and the pyridine-2-carboxylates (picloram, clopyralid, and aminopyralid). In the last 10 years, two novel pyridine-2-carboxylate (or picolinate) herbicides were discovered at Dow AgroSciences. This paper will describe the structure activity relationship study that led to the discovery of the 6-aryl-picolinate herbicides Arylex™ active (2005) and Rinskor™ active (2010). While Arylex was developed primarily for use in cereal crops and Rinskor is still in development primarily for use in rice crops, both herbicides will also be utilized in additional crops. |
| Databáze: | OpenAIRE |
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