Concomitant ring contraction cyclization strategy for the synthesis of novel 4-oxo-4,5-dihydro-pyrroloquinolines

Autor: Jean Paul Pradere, Stephane Sabelle, Hicham Bakkali, G. T. Manh, Muriel Pipelier, Remy Tuloup, Lucie Maingot, Didier Dubreuil, Uday Joshi
Rok vydání: 2004
Předmět:
Zdroj: Tetrahedron Letters. 45:5913-5916
ISSN: 0040-4039
DOI: 10.1016/j.tetlet.2004.05.115
Popis: The synthesis of novel substituted pyrroloquinolinones is described by concomitant ring contraction cyclization form 2-(2-amino-5-nitro-phenyl)-[4 H ]-1,3-thiazines, which were derived from N -substituted 5-nitro-anthranilonitrile. An easy access to novel 4-thiono-1,4-dihydro-1,3-quinazoline heterocycles is also mentioned.
Databáze: OpenAIRE