Copper(I) Oxide Catalyzed N-Arylation of Azoles and Amines with Arylboronic Acid at Room Temperature under Base-Free Conditions

Autor: Gopaladasu T. Venkanna, Kota Balaji Shiva Kumar, Bojja Sreedhar, V. Balasubrahmanyam
Rok vydání: 2008
Předmět:
Zdroj: Synthesis. 2008:795-799
ISSN: 1437-210X
0039-7881
DOI: 10.1055/s-2008-1032184
Popis: N -Arylation of azoles and amines with arylboronic acids was efficiently carried out with heterogeneous copper(I) oxide in methanol at room temperature under base-free conditions. The products N-arylazoles and N-arylamines were isolated in good to excellent yields. A variety of arylboronic acids and amines were converted to the corresponding N-arylazoles and N-arylamines, demonstrating the versatality of the reaction.
Databáze: OpenAIRE