Synthesis of 2-Aryl[1]benzofuro[2,3-e][1,2,4]triazin-3(2H)-ones and Their Use for Preparation of 1-Aryl-5-(2-hydroxyphenyl)-6-azauracils

Autor: Jakub Stýskala, Jan Slouka, Vojtěch Bekárek, Miloslav Hejsek
Rok vydání: 1997
Předmět:
Zdroj: Collection of Czechoslovak Chemical Communications. 62:1754-1762
ISSN: 1212-6950
0010-0765
Popis: A series of arylhydrazones 1a-1i was prepared by coupling of arene diazonium salts with ethyl N-(benzo[b]furan-2-yl)carbamate. The hydrazones 1 were thermally cyclized to the corresponding 2-aryl[1]benzofuro[2,3-e][1,2,4]triazin-3(2H)-ones 2a-2i, derivatives of a new fused ring system. Compounds 2 were transformed by hydrolytic splitting to the corresponding 1-aryl-5-(2-hydroxyphenyl)-6-azauracils 3a-3i.
Databáze: OpenAIRE