One-pot synthesis of 2-methyl-1,5-diaromatic-1H-pyrroles from styrene, acetone and arylamines using TBHP, copper(II) trifluoromethanesulfonate and sulfamic acid

Autor: Yufei Han, Shaowei Chen, Ping Gong, Dengzhi Xu, Zhenliang Shan, Liying Xu, Bingfu Zhang, Shimei Du, Congjun Xu
Rok vydání: 2018
Předmět:
Zdroj: Tetrahedron Letters. 59:260-263
ISSN: 0040-4039
DOI: 10.1016/j.tetlet.2017.12.031
Popis: The one-pot copper/manganese co-catalyzed heterocyclization of arylamine derivatives with styrene and acetone to produce a series of 2-methyl-1,5-diaromatic-1 H -pyrroles was investigated. The described reaction combines 1,4-dicarbonyl synthesis and Paal-Knorr type condensation reactions.
Databáze: OpenAIRE