TBHP/KI-Promoted Oxidative Cyclization of α-Aminoketones for One-Pot Synthesis of Substituted 2-Acyloxazoles
| Autor: | Zongjie Gan, Lin Ling Gan, Dali Zhu, Jiecheng Zheng, Zhangyou Yang, Huali Chen, Wei Wang |
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| Rok vydání: | 2022 |
| Předmět: | |
| Zdroj: | Synthesis. 55:1419-1426 |
| ISSN: | 1437-210X 0039-7881 |
| DOI: | 10.1055/a-1996-8388 |
| Popis: | A metal-free and facile synthesis of substituted 2-acyloxazole derivatives from α-aminoketones was developed via a TBHP/KI-promoted oxidative cyclization. This procedure proceeded smoothly under mild conditions and a broad scope of 2-acyloxazoles were obtained in moderate to good yields. |
| Databáze: | OpenAIRE |
| Externí odkaz: |
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