Cyclization of 1-acylaminoacridones into 7H-pyrido[2,3,4-kl]acridin-2(3H)-ones

Autor: S. P. Titova, M. V. Gorelik, E. V. Gordievskaya
Rok vydání: 2006
Předmět:
Zdroj: Russian Chemical Bulletin. 55:1487-1491
ISSN: 1573-9171
1066-5285
Popis: 1-Acylamino-10-methylacridones in a polar aprotic solvent underwent base-catalyzed cyclization into the corresponding 7-methyl-7H-pyrido[2,3,4-kl]acridin-2(3H)-ones. Heating of 1-butylaminoacridone in acetic anhydride in the presence of p-toluenesulfonic acid and potassium acetate afforded 3-butyl-7H-pyrido[2,3,4-kl]acridin-2(3H)-one, while heating of 1-aminoacridone under the same conditions gave 9-acetoxy-1-acetylimino-1,10-dihydroxy-acridine.
Databáze: OpenAIRE