Synthesis of a 6H-Pyrazolo[4,5,1-de]acridin-6-one Derivative: A Useful Intermediate of Antitumour Agents
Autor: | Yukiteru Mimura, Shinji Tomioka, Toru Sugaya, Takashi Mimura, Masanori Ikuta, Nobuyuki Kato, Masaji Fujisawa-shi Kasai |
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Rok vydání: | 1994 |
Předmět: | |
Zdroj: | Synthesis. 1994:73-76 |
ISSN: | 1437-210X 0039-7881 |
Popis: | A 6H-pyrazolo[4,5,1-de]acridin-6-one derivative, a useful intermediate of antitumor agents, was prepared by a facile synthetic route from 2-bromobenzoic acid and 6-nitroindazole involving a halogenocopper(I)-catalyzed Ullmann coupling reaction and Friedel-Crafts cyclization. |
Databáze: | OpenAIRE |
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