A Novel Method for N3-Functionalized Aminoimidazolines and Aminopyrimidines by Aza-Michael Additions of Aminoimidazolines and Aminopyrimidines to α,β-Unsaturated Carbonyl Compounds

Autor:	Chengwei Lv, Guo-Li Huang, Wen-Long Yang, Xicun Wang, Zheng-Jun Quan
Rok vydání:	2007
Předmět:	Pharmacology Chemistry Organic Chemistry Regioselectivity Combinatorial chemistry Analytical Chemistry Catalysis
Zdroj:	HETEROCYCLES. 71:2363
ISSN:	0385-5414
DOI:	10.3987/com-07-11118
Popis:	An efficient and convenient procedure is described for the preparation of N3-functionalized aminoimidazolines and aminopyrimidines through the aza-Michael additions of aminoimidazolines and aminopyrimidines with a, /?-unsaturated carbonyl compounds catalyzed by KF/Al 2 O 3 . This method offers a novel and efficient protocol for the N3-functionalized aminoimidazolines and aminopyrimidines with good regioselectivity and high purity under mild conditions.
Databáze:	OpenAIRE
Externí odkaz:	https://explore.openaire.eu/search/publication?articleId=doi_________::a512c9f51e296c7342ad98d8912ef2c3 https://doi.org/10.3987/com-07-11118 Zobrazit plný text záznamu