Phenylaziridine as a 1,3-dipole. Application to the synthesis of functionalized pyrrolidines

Autor:	André Mann, Ioana Ungureanu, Cristian Bologa, Said Chayer
Rok vydání:	1999
Předmět:	Chemistry Organic Chemistry Drug Discovery Organic chemistry Reactivity (chemistry) Lewis acids and bases Biochemistry Medicinal chemistry 1 3-dipole Ion
Zdroj:	Tetrahedron Letters. 40:5315-5318
ISSN:	0040-4039
DOI:	10.1016/s0040-4039(99)01002-3
Popis:	ce:simple-parahenylaziridine 1 in the presence of an appropriate Lewis acid reacts as a 1,3-dipole. The cyclocondensation of 1 with DHP in the presence of BF 3 ·Et 2 O produced the azaoxa[3.2.0] cycloadducts 4a–4b . The reactivity of the corresponding N -tosyliminium ions was explored.
Databáze:	OpenAIRE
Externí odkaz:	https://explore.openaire.eu/search/publication?articleId=doi_________::8f2960cc4dde9ac1f3daf9bd9c225319 https://doi.org/10.1016/s0040-4039(99)01002-3 Zobrazit plný text záznamu Full Text from ScienceDirect