Straightforward and mild deprotection methods of N-mono- and N,N-functionalised bisaminal cyclens

Autor:	Maryline Beyler, Raphaël Tripier, Fatima Oukhatar
Rok vydání:	2015
Předmět:	chemistry.chemical_classification chemistry.chemical_compound chemistry Cyclen Transamination Organic Chemistry Drug Discovery Organic chemistry Glyoxal Biochemistry Combinatorial chemistry Vicinal 3. Good health
Zdroj:	Tetrahedron. 71:3857-3862
ISSN:	0040-4020
DOI:	10.1016/j.tet.2015.04.021
Popis:	Strategic removal of the bisaminal bridge of N-mono- and N1,N7-difunctionalised cyclen glyoxal derivatives was carried out via transamination processes with vicinal diamines. These procedures were found to be particularly well-suited for cyclen targets bearing sensitive groups.
Databáze:	OpenAIRE
Externí odkaz:	https://explore.openaire.eu/search/publication?articleId=doi_________::8e751949b9dca00aa0735f36e66be36a https://doi.org/10.1016/j.tet.2015.04.021 Zobrazit plný text záznamu Full Text from ScienceDirect