Copper Acetate Aerobic Oxidative Synthesis of Pyrido[1,2-a]benzimidazoles from Aminopyridines and Phenylboronic Acids

Autor: Xiao-Qiang Zhou, Shuan Zhang, Guanghui Zhang, Hao Yan, Zhenyu Zuo, Hui Guo, Jingli Liu
Rok vydání: 2019
Předmět:
Zdroj: Synlett. 30:1469-1473
ISSN: 1437-2096
0936-5214
DOI: 10.1055/s-0037-1611847
Popis: Pyrido[1,2-a]benzimidazoles, which show interesting and potentially useful biological activities, have drawn extensive attention from chemists. A straightforward copper acetate-oxidative one-pot synthesis of these compounds from 2-aminopyridines and phenylboronic acids through C–N bond formation and C–H bond activation was developed as a simple and convenient method.
Databáze: OpenAIRE