Synthesis and fungicidal activity ofN-(p-sulfonylphenyl)-N1 -carbamoylureas

Autor: Richard M. Ellam, Sultan Farouk, Richard J. Cremlyn
Rok vydání: 1998
Předmět:
Zdroj: Pesticide Science. 52:70-74
ISSN: 0031-613X
DOI: 10.1002/(sici)1096-9063(199801)52:1<70::aid-ps668>3.0.co;2-f
Popis: A series of 11 N-(p-sulfonylphenyl)-N 1 -carbamoylureas was prepared by reaction of 1,6-diphenyl-2,4-dioxohexahydro-s-triazine with chlorosulfonic acid and thionyl chloride. The resultant N-(p-chlorosulfonylphenyl)-N 1 -carbamoylurea was subsequently condensed with amines, butanol, hydrazine and sodium azide. The hydrazide was reacted with carbonyl compounds and the azide with trimethyl phosphite. The products were tested for in-vivo fungicidal activity against barley powdery mildew (Erysiphe graminis); the acetone hydrazone derivative showed the highest activity.
Databáze: OpenAIRE