Synthesis of 4,5,6,7-tetrahydrobenzoxazol-2-ones by a highly regioselective Diels-Alder cycloaddition of exo-oxazolidin-2-one dienes with chalcones

Autor:	Joaquín Tamariz, Aydeé Fuentes-Benítes, Salvador Mastachi-Loza, Eduardo Díaz-Torres, Asenet Tapia-Bustamante, Rubén A. Toscano, Tania I. Ramírez-Candelero, Carlos González-Romero
Rok vydání:	2019
Předmět:	Chalcone 010405 organic chemistry Organic Chemistry Regioselectivity 010402 general chemistry 01 natural sciences Biochemistry Cycloaddition 0104 chemical sciences chemistry.chemical_compound chemistry Drug Discovery Diels alder Organic chemistry Stereoselectivity Diels–Alder reaction
Zdroj:	Tetrahedron Letters. 60:1370-1374
ISSN:	0040-4039
Popis:	The synthesis of novel of 4,5,6,7-tetrahydrobenzoxazol-2-ones is herein reported. They were obtained in moderate to good yields by a highly regio- and stereoselective Diels-Alder cycloaddition of N-substituted exo-oxazolidin-2-one dienes with chalcones or bis-chalcones as dienophiles.
Databáze:	OpenAIRE
Externí odkaz:	https://explore.openaire.eu/search/publication?articleId=doi_________::7b118b0835732cc6e5d1f5497d30e4bf https://doi.org/10.1016/j.tetlet.2019.04.027 Zobrazit plný text záznamu Full Text from ScienceDirect