Cu-Mediated Expeditious Annulation of Alkyl 3-Aminoacrylates with Aryldiazonium Salts: Access to Alkyl N2-Aryl 1,2,3-Triazole-carboxylates for Druglike Molecular Synthesis

Autor:	Hao-Nan Liu, Hao-Qiang Cao, Jun-An Ma, Chi Wai Cheung
Rok vydání:	2020
Předmět:	chemistry.chemical_classification Annulation 1 2 3-Triazole 010405 organic chemistry Aryl Organic Chemistry 010402 general chemistry 01 natural sciences Biochemistry 0104 chemical sciences chemistry.chemical_compound chemistry Molecule Organic chemistry Physical and Theoretical Chemistry Alkyl
Zdroj:	Organic Letters. 22:1396-1401
ISSN:	1523-7052 1523-7060
DOI:	10.1021/acs.orglett.0c00006
Popis:	Alkyl N-aryl 1,2,3-triazole-carboxylates are important molecules or intermediates in medicinal chemistry, but the synthesis of N2-aryl counterparts remains elusive. Herein, we describe a Cu-mediate...
Databáze:	OpenAIRE
Externí odkaz:	https://explore.openaire.eu/search/publication?articleId=doi_________::722e070368e6a5882582a00a0af1f4b5 https://doi.org/10.1021/acs.orglett.0c00006 Zobrazit plný text záznamu