ChemInform Abstract: An Intramolecular C-N Cross-Coupling of β-Enaminones: A Simple and Efficient Way to Precursors of Some Alkaloids of Galipea officinalis
Autor: | Hana Doušová, Radim Horak, Petr Simunek, Zdenka Ruzickova |
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Rok vydání: | 2015 |
Předmět: | |
Zdroj: | ChemInform. 46 |
ISSN: | 0931-7597 |
DOI: | 10.1002/chin.201532167 |
Popis: | A simple and efficient method for the intramolecular, palladium catalyzed amination of both chloro- and bromo-substituted 3-amino-1,5-diphenylpent-2-en-1-ones (I) is developed furnishing 2-aroylmethylidene-1,2,3,4-tetrahydroquinolines (II) as suitable precursors for the synthesis of alkaloids from Galipea officinalis. |
Databáze: | OpenAIRE |
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