ChemInform Abstract: An Intramolecular C-N Cross-Coupling of β-Enaminones: A Simple and Efficient Way to Precursors of Some Alkaloids of Galipea officinalis

Autor: Hana Doušová, Radim Horak, Petr Simunek, Zdenka Ruzickova
Rok vydání: 2015
Předmět:
Zdroj: ChemInform. 46
ISSN: 0931-7597
DOI: 10.1002/chin.201532167
Popis: A simple and efficient method for the intramolecular, palladium catalyzed amination of both chloro- and bromo-substituted 3-amino-1,5-diphenylpent-2-en-1-ones (I) is developed furnishing 2-aroylmethylidene-1,2,3,4-tetrahydroquinolines (II) as suitable precursors for the synthesis of alkaloids from Galipea officinalis.
Databáze: OpenAIRE