Synthesis of substituted fused pyridines, pyrazines and pyrimidines by sequential Ugi/inverse electron demand Diels–Alder transformations

Autor: Irini Akritopoulou-Zanze, Hongyu Zhao, Ying Wang, Stevan W. Djuric
Rok vydání: 2009
Předmět:
Zdroj: Tetrahedron Letters. 50:5773-5776
ISSN: 0040-4039
Popis: The synthesis of all four regioisomers of fused pyrrolidino-pyridines in a one-pot two-step sequential Ugi-inverse electron demand Diels–Alder reaction is described. Fused pyrrolidino-pyrazines, pyrrolidino-pyrimidines and azepinone pyridines can also be obtained in consecutive synthetic sequences.
Databáze: OpenAIRE