Synthesis of 1,5-Disubstituted Tetrazoles from Nitrones by Using Bis(p-nitrophenyl) Phosphorazidate in the Presence of 4-(Dimethylamino)pyridine

Autor:	Masato Matsugi, Kotaro Ishihara, Takayuki Shioiri
Rok vydání:	2022
Předmět:	Organic Chemistry
Zdroj:	Synlett. 33:781-784
ISSN:	1437-2096 0936-5214
DOI:	10.1055/a-1800-2011
Popis:	A novel method has been developed for the synthesis of 1,5-disubstituted tetrazoles from nitrones by using bis(p-nitrophenyl) phosphorazidate in the presence of 4-(dimethylamino)pyridine. By this approach, various nitrones were converted into the corresponding tetrazoles. This method permits the preparation of 1,5-disubstituted tetrazoles without the need for toxic or explosive reagents.
Databáze:	OpenAIRE
Externí odkaz:	https://explore.openaire.eu/search/publication?articleId=doi_________::4715fb3470b63be0647f475cca67939e https://doi.org/10.1055/a-1800-2011 Zobrazit plný text záznamu