ChemInform Abstract: α-Azido Acids in Heterocyclic Synthesis

Autor: Steven W. Goldstein, Ruth E. McDermott, Michael Raymond Makowski, Cynthia Eller
Rok vydání: 2010
Předmět:
Zdroj: ChemInform. 23
ISSN: 0931-7597
DOI: 10.1002/chin.199225192
Popis: 2-Aminobenzophenones and acetophenones were N-acylated with α-azido carboxylic acids to give the corresponding anilides. Reductive cyclization provided 3-substituted-2H-1,4-benzodiazepin-2-ones in good (46–99%) yields.
Databáze: OpenAIRE