ChemInform Abstract: α-Azido Acids in Heterocyclic Synthesis
Autor: | Steven W. Goldstein, Ruth E. McDermott, Michael Raymond Makowski, Cynthia Eller |
---|---|
Rok vydání: | 2010 |
Předmět: | |
Zdroj: | ChemInform. 23 |
ISSN: | 0931-7597 |
DOI: | 10.1002/chin.199225192 |
Popis: | 2-Aminobenzophenones and acetophenones were N-acylated with α-azido carboxylic acids to give the corresponding anilides. Reductive cyclization provided 3-substituted-2H-1,4-benzodiazepin-2-ones in good (46–99%) yields. |
Databáze: | OpenAIRE |
Externí odkaz: |