Copper-Catalyzed Synthesis of β- and δ-Carbolines by Double N-Arylation of Primary Amines
Autor: | Nguyen Ngoc Tuan, Hoang Le Tuan Anh, Nguyen Van Tuyen, Peter Langer, Tuan Thanh Dang, Ha Nam Do, Nguyen Minh Quan, Tran Quang Hung, Ban Van Phuc, Nguyen Quang An |
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Rok vydání: | 2021 |
Předmět: | |
Zdroj: | Synlett. 32:1004-1008 |
ISSN: | 1437-2096 0936-5214 |
DOI: | 10.1055/s-0040-1720461 |
Popis: | Two efficient and practical approaches are reported for the synthesis of β- and δ-carbolines from 3,4-dibromopyridine. The synthesis is based on site-selective Cu-catalyzed double C–N coupling reactions and subsequent annulations by twofold Pd-catalyzed C–N coupling with amines. |
Databáze: | OpenAIRE |
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